Targacept, Inc.

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Patent Activity in the Last 10 Years

Technologies

Intl Class Technology Matters Rank in Class
 
 
 
A61K PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES 23232
 
 
 
C07D HETEROCYCLIC COMPOUNDS 15147
 
 
 
A61P THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS 544
 
 
 
A01N PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF 392
 
 
 
C07C ACYCLIC OR CARBOCYCLIC COMPOUNDS 1137
 
 
 
C12N MICRO-ORGANISMS OR ENZYMES; COMPOSITIONS THEREOF 1166

Top Patents (by citation)

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Recent Publications

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Recent Patents

Patent # Title Filing Date Issue Date Intl Class
9532974 Nicotinic receptor non-competitive antagonistsAug 27, 15Jan 03, 17[A61K, C07D, C07C]
9107915 Hydroxybenzoate salts of metanicotine compoundsJun 05, 14Aug 18, 15[A61K, C07D]
8901177 Method of treating bladder disordersMar 13, 13Dec 02, 14[A61K]
8809397 Nicotinic receptor non-competitive antagonistsMay 24, 11Aug 19, 14[A61K, C07C]
8802694 3,6-diazabicyclo[3.1.1]heptanes as neuronal nicotinic acetycholine receptor ligandsDec 03, 10Aug 12, 14[A61K, C07D]
8778978 Hydroxybenzoate salts of metanicotine compoundsOct 03, 13Jul 15, 14[A61K]
8703802 Process for the preparation of aryl substituted olefinic aminesMay 19, 11Apr 22, 14[A61K, A01N, C07D]
8633227 Synthesis and novel salt forms of (R)-3-((E)-pyrrolidin-3-yl)vinyl)-5-tetrahydropyran-4-yloxy)pyridineNov 30, 09Jan 21, 14[A61K, C07D]
8053451 Hydroxybenzoate salts of metanicotine compoundsNov 04, 08Nov 08, 11[A61K, A01N, C07D]
7790757 Compounds capable of activating cholinergic receptorsOct 31, 07Sep 07, 10[A61K, C07D, A61P]

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Expired/Abandoned/Withdrawn Patents

Patent # Title Status Filing Date Issue/Pub Date Intl Class
2014/0288,169 NICOTINIC RECEPTOR NON-COMPETITIVE ANTAGONISTSAbandonedJan 05, 12Sep 25, 14[C07D, C07C]
2014/0288,185 NICOTINIC RECEPTOR NON-COMPETITIVE MODULATORSAbandonedNov 01, 12Sep 25, 14[C07C]
2014/0249,141 1,4-DIAZABICYCLO[3.2.2]NONANES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDSAbandonedAug 20, 12Sep 04, 14[A61K, C07D]
2014/0234,270 TREATMENT WTH ALPHAT SELECTIVE LIGANDSAbandonedApr 23, 14Aug 21, 14[A61K]
2014/0024,638 TREATMENT OF COGNITIVE DYSFUNCTION IN SCHIZOPHRENIAAbandonedJan 17, 12Jan 23, 14[A61K]
2013/0310,425 NOVEL POLYMORPH FORMS OF (2S)-(4E)-N-METHYL-5-[3-(5-ISOPROPOXYPYRIDIN)YL]-4-PENTEN-2-AMINEAbandonedMay 14, 13Nov 21, 13[C07D]
8580826 Hydroxybenzoate salts of metanicotine compoundsExpiredOct 26, 11Nov 12, 13[A61K, C07D, A61P]
2013/0237,550 ARYLVINYLAZACYCLOALKANE COMPOUNDS FOR CONSTIPATIONAbandonedMar 04, 11Sep 12, 13[A61K]
8461344 Polymorph forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropdxypyridin)yl]-4-penten-2-amineExpiredMay 08, 07Jun 11, 13[A61K, C07D]
8288420 Compounds capable of activating cholinergic receptorsExpiredMay 10, 10Oct 16, 12[A61K, C07D, A61P]
2012/0190,752 EXO-S-MECAMYLAMINE METHOD, USE, AND COMPOUND FOR TREATMENTAbandonedJul 12, 10Jul 26, 12[A61K, A61P]
2012/0157,477 REVERSAL OF L-DOPA-INDUCED DYSKINESIA BY NEURONAL NICOTINIC RECEPTOR LIGANDSAbandonedJun 15, 10Jun 21, 12[A61K, A61P]
8198296 Sub-type selective azabicycloalkane derivativesExpiredMar 27, 08Jun 12, 12[A61K, C07D]
2012/0053,168 FUSED BENZOAZEPINES AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDSAbandonedFeb 16, 10Mar 01, 12[A61K, C07D, A61P]
2011/0262,407 TREATMENT WITH ALPHA7 SELECTIVE LIGANDSAbandonedNov 09, 09Oct 27, 11[A61K, A61P]
2011/0263,629 AMIDES OF DIAZABICYCLOOCTANES AND USES THEREOFAbandonedSep 02, 09Oct 27, 11[A61K, C07D, A61P]
2011/0257,168 DERIVATIVES OF OXABISPIDINE AS NEURONAL NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDSAbandonedJul 01, 09Oct 20, 11[A61K, C07D, A61P]
8017785 Salt forms of (2S)-(4E)-N-methyl-5-[3-(5-isopropoxypyridin)y1]-4-penten 2-amineExpiredMay 08, 07Sep 13, 11[A61P]
2011/0124,678 TREATMENT WITH ALPHA 7-SELECTIVE LIGANDSAbandonedAug 01, 08May 26, 11[A61K, C07D, A61P]
2011/0118,239 PREPARATION AND ENANTIOMERIC SEPARATION OF 7-(3-PYRIDINYL)-1,7-DIAZASPIRO[4.4]NONANE AND NOVEL SALT FORMS OF THE RACEMATE AND ENANTIOMERSAbandonedJan 15, 09May 19, 11[A61K, C07D, A61P]

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